Names and pronunciation
(rip-re′ti-nib) Qinlock
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Drug reference
(rip-re′ti-nib) Qinlock
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Func. class.: Antineoplastic, tyrosine kinase inhibitor
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USES: Treatment of advanced gastrointestinal stromal tumor (GIST) in those who have received ≥3 kinase inhibitors, including imatinib
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CONTRAINDICATIONS: Hypersensitivity, pregnancy, breastfeeding
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DOSAGE AND ROUTES Adult: PO 150 mg daily until disease progression or unacceptable toxicity
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Available forms: Tablet 50 mg
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